Researcher Portfolio
Offermanns, Stefan
Pharmacology, Max Planck Institute for Heart and Lung Research, Max Planck Society
Researcher Profile
Position: Pharmacology, Max Planck Institute for Heart and Lung Research, Max Planck Society
Researcher ID: https://pure.mpg.de/cone/persons/resource/persons224185
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Publications
(1 - 25 of 166)
: Kwon, J., Haruya, K., Mattonet, K., Guenther, S., Hahnefeld, L., Shamsara, J., Heering, J., Kurz, M., Kirchhofer, S., Krasel, C., Ulrich, M., Persechino, M., Murthy, S., Orlandi, C., Sadik, C. D., Geisslinger, G., Buenemann, M., Kolb, P., Offermanns, S., & Wettschureck, N. (2025). Orphan G protein-coupled receptor GPRC5B controls macrophage function by facilitating prostaglandin E receptor 2 signaling. NATURE COMMUNICATIONS, 16(1): 1448. doi:10.1038/s41467-025-56713-0. [PubMan] : Jin, Y.-J., Liang, G., Li, R., Wang, S., Alnouri, M. W., Bentsen, M., Kuenne, C., Guenther, S., Yan, Y., Li, Y., Wettschureck, N., & Offermanns, S. (2025). Phosphorylation of endothelial histone H3.3 serine 31 by PKN1 links flow-induced signaling to proatherogenic gene expression. NATURE CARDIOVASCULAR RESEARCH, 4(2). doi:10.1038/s44161-024-00593-y. [PubMan] : Su, M., Zhao, W., Jiang, H., Zhao, Y., Liao, Z., Liu, Z., Xu, M., Jiang, S., Wu, L., Yang, Y., Wang, Z., Zeng, Z., Fang, Y., Tang, C., Miller, C. L., Evans, P. C., Wang, L., Banach, M., Jo, H., Berk, B. C., Offermanns, S., Huang, Y., Ge, J., Xu, S., & Weng, J. (2025). Endothelial IGFBP6 suppresses vascular inflammation and atherosclerosis. NATURE CARDIOVASCULAR RESEARCH, 4(2). doi:10.1038/s44161-024-00591-0. [PubMan] : Hernandez-Olmos, V., Heering, J., Ildefeld, N., Ehrler, J. H. M., Kaps, A., Rajkumar, R., Marinescu, B., Kaiser, A., Macinkovic, I., Elewa, M. A. F., Alnouri, M. W., Elson, L., Schubert-Zsilavecz, M., Kallenborn-Gerhardt, W., Schmidtko, A., Mueller, S., Offermanns, S., Steinhilber, D., Weigert, A., & Proschak, E. (2025). Identification of a Chemical Probe for BLT2 Activation by Scaffold Hopping. JOURNAL OF MEDICINAL CHEMISTRY, 68(2), 1195-1221. doi:10.1021/acs.jmedchem.4c01617. [PubMan] : Yoshida, T., Yoshida, S., Inukai, K., Kato, K., Yura, Y., Hattori, T., Taki, K., Enomoto, A., Ohashi, K., Okumura, T., Ouchi, N., Kawase, H., Wettschureck, N., Offermanns, S., Murohara, T., & Takefuji, M. (2024). ALPK2 prevents cardiac diastolic dysfunction in heart failure with preserved ejection fraction. FASEB JOURNAL, 38(22): e70192. doi:10.1096/fj.202402103R. [PubMan] : Alnouri, M. W., Roquid, K. A., Bonnavion, R., Cho, H., Heering, J., Kwon, J., Jaeger, Y., Wang, S., Guenther, S., Wettschureck, N., Geisslingerb, G., Gurke, R., Mueller, C. E., Proschak, E., & Offermanns, S. (2024). SPMs exert anti- inflammatory and pro- resolving effects through positive allosteric modulation of the prostaglandin EP4 receptor. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 121(41): e2407130121. doi:10.1073/pnas.2407130121. [PubMan] : Yoshida, S., Yoshida, T., Inukai, K., Kato, K., Yura, Y., Hattori, T., Enomoto, A., Ohashi, K., Okumura, T., Ouchi, N., Kawase, H., Wettschureck, N., Offermanns, S., Murohara, T., & Takefuji, M. (2024). Protein kinase N promotes cardiac fibrosis in heart failure by fibroblast-to-myofibroblast conversion. NATURE COMMUNICATIONS, 15(1): 7638. doi:10.1038/s41467-024-52068-0. [PubMan] : Keshavarz, M., Ruppert, A.-L., Meiners, M., Poharkar, K., Liu, S., Mahmoud, W., Winterberg, S., Hartmann, P., Mermer, P., Perniss, A., Offermanns, S., Kummer, W., & Schuetz, B. (2024). Bitter tastants relax the mouse gallbladder smooth muscle independent of signaling through tuft cells and bitter taste receptors. SCIENTIFIC REPORTS, 14(1): 18447. doi:10.1038/s41598-024-69287-6. [PubMan] : Peng, Y., Du, J., Li, R., Guenther, S., Wettschureck, N., Offermanns, S., Wang, Y., Schneider, A., & Braun, T. (2024). RhoA-mediated G12-G13 signaling maintains muscle stem cell quiescence and prevents stem cell loss. CELL DISCOVERY, 10(1): 76. doi:10.1038/s41421-024-00696-7. [PubMan] : Hernandez-Olmos, V., Heering, J., Marinescu, B., Schermeng, T., Ivanov, V. V., Moroz, Y. S., Nevermann, S., Mathes, M., Ehrler, J. H. M., Alnouri, M. W., Wolf, M., Haydo, A. S., Schmachtel, T., Zaliani, A., Ho''fner, G., Kaiser, A., Schubert-Zsilavecz, M., Beck-Sickinger, A. G., Offermanns, S., Gribbon, P., Rieger, M. A., Merk, D., Sisignano, M., Steinhilber, D., & Proschak, E. (2024). Development of a Potent and Selective G2A (GPR132) Agonist. JOURNAL OF MEDICINAL CHEMISTRY. doi:10.1021/acs.jmedchem.3c02164. [PubMan] : Wang, T., Shao, J., Shamit, K., Alnouri, M. W., Carvalho, J., Guenther, S., Krasel, C., Murphy, K. T., Buenemann, M., Offermanns, S., & Wettschureck, N. (2024). Orphan GPCR GPRC5C Facilitates Angiotensin II-Induced Smooth Muscle Contraction. CIRCULATION RESEARCH, 134(10), 1259-1275. doi:10.1161/CIRCRESAHA.123.323752. [PubMan] : Wu, F., Li, X., Looso, M., Liu, H., Ding, D., Guenther, S., Kuenne, C., Liu, S., Weissmann, N., Boettger, T., Atzberger, A., Kolahian, S., Renz, H., Offermanns, S., Gaertner, U., Potente, M., Zhou, Y., Yuan, X., & Braun, T. (2024). Spurious transcription causing innate immune responses is prevented by 5-hydroxymethylcytosine. NATURE GENETICS, 55(1), 100-+. doi:10.1038/s41588-022-01252-3. [PubMan] : Trif, C., Banica, A.-M., Manolache, A., Anghel, S. A., Hutanu, D.-E., Stratulat, T., Badea, R., Oprita, G., Selescu, T., Petrescu, S. M., Sisignano, M., Offermanns, S., Babes, A., & Tunaru, S. (2023). Inhibition of TRPM8 function by prostacyclin receptor agonists requires coupling to Gq/11 proteins. BRITISH JOURNAL OF PHARMACOLOGY. doi:10.1111/bph.16295. [PubMan] : Balla, H., Borsodi, K., Orsy, P., Horvath, B., Molnar, P. J., Lenart, A., Kosztelnik, M., Ruisanchez, E., Wess, J., Offermanns, S., Nyirady, P., & Benyo, Z. (2023). Intracellular signaling pathways of muscarinic acetylcholine receptor-mediated detrusor muscle contractions. AMERICAN JOURNAL OF PHYSIOLOGY-RENAL PHYSIOLOGY, 325(5), F618-F628. doi:10.1152/ajprenal.00261.2022. [PubMan] : Balla, H., Borsodi, K., Orsy, P., Horvath, B., Molnar, P. J., Lenart, A., Kosztelnik, M., Ruisanchez, E., Wess, J., Offermanns, S., Nyirady, P., & Benyo, Z. (2023). Intracellular signaling pathways of muscarinic acetylcholine receptor-mediated detrusor muscle contractions. AMERICAN JOURNAL OF PHYSIOLOGY-RENAL PHYSIOLOGY, 325(5), F618-F628. doi:10.1152/ajprenal.00261.2022. [PubMan] : Bonnavion, R., Liu, S., Kawase, H., Roquid, K. A., & Offermanns, S. (2023). Large chemokine binding spectrum of human and mouse atypical chemokine receptor GPR182 (ACKR5). FRONTIERS IN PHARMACOLOGY, 14: 1297596. doi:10.3389/fphar.2023.1297596. [PubMan] : Alexander, S. P. H., Mathie, A. A., Peters, J. A., Veale, E. L., Striessnig, J., Kelly, E., Armstrong, J. F., Faccenda, E., Harding, S. D., Davies, J. A., Aldrich, R. W., Attali, B., Baggetta, A. M., Becirovic, E., Biel, M., Bill, R. M., Caceres, A. I., Catterall, W. A., Conner, A. C., Davies, P., De Clerq, K., Delling, M., Di Virgilio, F., Falzoni, S., Fenske, S., Fortuny-Gomez, A., Fountain, S., George, C., Goldstein, S. A. N., Grimm, C., Grissmer, S., Ha, K., Hammelmann, V., Hanukoglu, I., Hu, M., Ijzerman, A. P., Jabba, S. V., Jarvis, M., Jensen, A. A., Jordt, S. E., Kaczmarek, L. K., Kellenberger, S., Kennedy, C., King, B., Kitchen, P., Liu, Q., Lynch, J. W., Meades, J., Mehlfeld, V., Nicke, A., Offermanns, S., Perez-Reyes, E., Plant, L. D., Rash, L., Ren, D., Salman, M. M., Sieghart, W., Sivilotti, L. G., Smart, T. G., Snutch, T. P., Tian, J., Trimmer, J. S., Van den Eynde, C., Vriens, J., Wei, A. D., Winn, B. T., Wulff, H., Xu, H., Yang, F., Fang, W., Yue, L., Zhang, X., & Zhu, M. (2023). The Concise Guide to PHARMACOLOGY 2023/24: Ion channels. BRITISH JOURNAL OF PHARMACOLOGY, 180, S145-S222. doi:10.1111/bph.16178. [PubMan] : Alexander, S. P. H., Christopoulos, A., Davenport, A. P., Kelly, E., Mathie, A. A., Peters, J. A., Veale, E. L., Armstrong, J. F., Faccenda, E., Harding, S. D., Davies, J. A., Abbracchio, M. P., Abraham, G., Agoulnik, A., Alexander, W., Al-hosaini, K., Baeck, M., Baker, J. G., Barnes, N. M., Bathgate, R., Beaulieu, J.-M., Beck-Sickinger, A. G., Behrens, M., Bernstein, K. E., Bettler, B., Birdsall, N. J. M., Blaho, V., Boulay, F., Bousquet, C., Braeuner-Osborne, H., Burnstock, G., Calo, G., Castano, J. P., Catt, K. J., Ceruti, S., Chazot, P., Chiang, N., Chini, B., Chun, J., Cianciulli, A., Civelli, O., Clapp, L. H., Couture, R., Cox, H. M., Csaba, Z., Dahlgren, C., Dent, G., Douglas, S. D., Dournaud, P., Eguchi, S., Escher, E., Filardo, E. J., Fong, T., Fumagalli, M., Gainetdinov, R. R., Garelja, M. L., de Gasparo, M., Gerard, C., Gershengorn, M., Gobeil, F., Goodfriend, T. L., Goudet, C., Graetz, L., Gregory, K. J., Gundlach, A. L., Hamann, J., Hanson, J., Hauger, R. L., Hay, D. L., Heinemann, A., Herr, D., Hollenberg, M. D., Holliday, N. D., Horiuchi, M., Hoyer, D., Hunyady, L., Husain, A., Ijzerman, A. P., Inagami, T., Jacobson, K. A., Jensen, R. T., Jockers, R., Jonnalagadda, D., Karnik, S., Kaupmann, K., Kemp, J., Kennedy, C., Kihara, Y., Kitazawa, T., Kozielewicz, P., Kreienkamp, H.-J., Kukkonen, J. P., Langenhan, T., Larhammar, D., Leach, K., Lecca, D., Lee, J. D., Leeman, S. E., Leprince, J., Li, X. X., Lolait, S. J., Lupp, A., Macrae, R., Maguire, J., Malfacini, D., Mazella, J., Mcardle, C. A., Melmed, S., Michel, M. C., Miller, L. J., Mitolo, V., Mouillac, B., Mueller, C. E., Murphy, P. M., Nahon, J.-L., Ngo, T., Norel, X., Nyimanu, D., O'Carroll, A.-M., Offermanns, S., Panaro, M. A., Parmentier, M., Pertwee, R. G., Pin, J.-P., Prossnitz, E. R., Quinn, M., Ramachandran, R., Ray, M., Reinscheid, R. K., Rondard, P., Rovati, G. E., Ruzza, C., Sanger, G. J., Schoeneberg, T., Schulte, G., Schulz, S., Segaloff, D. L., Serhan, C. N., Singh, K. D., Smith, C. M., Stoddart, L. A., Sugimoto, Y., Summers, R., Tan, V. P., Thal, D., Thomas, W. (. W., Timmermans, P. B. M. W. M., Tirupula, K., Toll, L., Tulipano, G., Unal, H., Unger, T., Valant, C., Vanderheyden, P., Vaudry, D., Vaudry, H., Vilardaga, J.-P., Walker, C. S., Wang, J. M., Ward, D. T., Wester, H.-J., Willars, G. B., Williams, T. L., Woodruff, T. M., Yao, C., & Ye, R. D. (2023). The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors. BRITISH JOURNAL OF PHARMACOLOGY, 180(2), S23-S144. doi:10.1111/bph.16177. [PubMan] : Goodwin, A. T., John, A. E., Joseph, C., Habgood, A., Tatler, A. L., Susztak, K., Palmer, M., Offermanns, S., Henderson, N. C., & Jenkins, R. G. (2023). Stretch regulates alveologenesis and homeostasis via mesenchymal G(alpha q/11)-mediated TGF beta 2 activation. DEVELOPMENT, 150(9): dev201046. doi:10.1242/dev.201046. [PubMan] : Li, R., Shao, J., Jin, Y. J., Haruya, K., Ong, Y. T., Troidl, K., Quan, Q., Wang, L., Bonnavion, R., Wietelmann, A., Helmbacher, F., Potente, M., Graumann, J., Wettschureck, N., & Offermanns, S. (2023). Endothelial FAT1 inhibits angiogenesis by controlling YAP/TAZ protein degradation via E3 ligase MIB2. NATURE COMMUNICATIONS, 14(1): 1980. doi:10.1038/s41467-023-37671-x. [PubMan] : Shorning, B., Trent, N., Griffiths, D. F., Worzfeld, T., Offermanns, S., Smalley, M. J., & Williamson, M. (2023). Plexin-B1 Mutation Drives Metastasis in Prostate Cancer Mouse Models. CANCER RESEARCH COMMUNICATIONS, 3(3), 444-458. doi:10.1158/2767-9764.CRC-22-0480. [PubMan] : Nakayama, A., Roquid, K. A., Iring, A., Strilic, B., Guenther, S., Chen, M., Weinstein, L. S., & Offermanns, S. (2023). Suppression of CCL2 angiocrine function by adrenomedullin promotes tumor growth. JOURNAL OF EXPERIMENTAL MEDICINE, 220(1): e20211628. doi:10.1084/jem.20211628. [PubMan] : Wu, F., Li, X., Looso, M., Liu, H., Ding, D., Guenther, S., Kuenne, C., Liu, S., Weissmann, N., Boettger, T., Atzberger, A., Kolahian, S., Renz, H., Offermanns, S., Gaertner, U., Potente, M., Zhou, Y., Yuan, X., & Braun, T. (2023). Spurious transcription causing innate immune responses is prevented by 5-hydroxymethylcytosine. NATURE GENETICS, (2023; 55(1)), 100-111. doi:10.1038/s41588-022-01252-3. [PubMan] : Manta, C.-P., Leibing, T., Friedrich, M., Nolte, H., Adrian, M., Schledzewski, K., Krzistetzko, J., Kirkamm, C., David Schmid, C., Xi, Y., Stojanovic, A., Tonack, S., de la Torre, C., Hammad, S., Offermanns, S., Krueger, M., Cerwenka, A., Platten, M., Goerdt, S., & Geraud, C. (2022). Targeting of Scavenger Receptors Stabilin-1 and Stabilin-2 Ameliorates Atherosclerosis by a Plasma Proteome Switch Mediating Monocyte/Macrophage Suppression. CIRCULATION, 146(23), 1783-1799. doi:10.1161/CIRCULATIONAHA.121.058615. [PubMan] : Wedel, S., Hahnefeld, L., Alnouri, M. W., Offermanns, S., Hausch, F., Geisslinger, G., & Sisignano, M. (2022). The FKBP51 Inhibitor SAFit2 Restores the Pain-Relieving C16 Dihydroceramide after Nerve Injury. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23(22): 14274. doi:10.3390/ijms232214274. [PubMan]