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Free keywords:
COPPER-MEDIATED FLUORINATION; ARYL FLUORIDES; CATALYZED FLUORINATION; NUCLEOPHILIC FLUORINATION; REDUCTIVE ELIMINATION; FUNCTIONALIZED ARYL; BOND FORMATION; CONVERSION; STANNANES; ALCOHOLS
Abstract:
We report a practical synthesis method of the reagent PhenoFluor on decagram scale, provide a new formulation of PhenoFluor as a toluene solution, which should decrease challenges associated with the moisture sensitivity of the reagent, and expand the substrate scope of deoxyfluorination with PhenoFluor to heteroaromatics.