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  THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors

Alexander, S. P. H., Christopoulos, A., Davenport, A. P., Kelly, E., Mathie, A., Peters, J. A., et al. (2021). THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors. BRITISH JOURNAL OF PHARMACOLOGY, 178(Supplement 1), S27-S156. doi:10.1111/bph.15538.

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Alexander, Stephen P. H., Author
Christopoulos, Arthur, Author
Davenport, Anthony P., Author
Kelly, Eamonn, Author
Mathie, Alistair, Author
Peters, John A., Author
Veale, Emma L., Author
Armstrong, Jane F., Author
Faccenda, Elena, Author
Harding, Simon D., Author
Pawson, Adam J., Author
Southan, Christopher, Author
Davies, Jamie A., Author
Abbracchio, Maria Pia, Author
Alexander, Wayne, Author
Al-hosaini, Khaled, Author
Baeck, Magnus, Author
Barnes, Nicholas M., Author
Bathgate, Ross, Author
Beaulieu, Jean-Martin, Author
Bernstein, Kenneth E., AuthorBettler, Bernhard, AuthorBirdsall, Nigel J. M., AuthorBlaho, Victoria, AuthorBoulay, Francois, AuthorBousquet, Corinne, AuthorBraeuner-Osborne, Hans, AuthorBurnstock, Geoffrey, AuthorCalo, Girolamo, AuthorCastano, Justo P., AuthorCatt, KevinJ, AuthorCeruti, Stefania, AuthorChazot, Paul, AuthorChiang, Nan, AuthorChini, Bice, AuthorChun, Jerold, AuthorCianciulli, Antonia, AuthorCivelli, Olivier, AuthorClapp, Lucie H., AuthorCouture, Rejean, AuthorCsaba, Zsolt, AuthorDahlgren, Claes, AuthorDent, Gordon, AuthorSingh, Khuraijam Dhanachandra, AuthorDouglas, Steven D., AuthorDournaud, Pascal, AuthorEguchi, Satoru, AuthorEscher, Emanuel, AuthorFilardo, Edward J., AuthorFong, Tung, AuthorFumagalli, Marta, AuthorGainetdinov, Raul R., Authorde Gasparo, Marc, AuthorGerard, Craig, AuthorGershengorn, Marvin, AuthorGobeil, Fernand, AuthorGoodfriend, Theodore L., AuthorGoudet, Cyril, AuthorGregory, Karen J., AuthorGundlach, Andrew L., AuthorHamann, Joerg, AuthorHanson, Julien, AuthorHauger, Richard L., AuthorHay, Debbie L., AuthorHeinemann, Akos, AuthorHollenberg, Morley D., AuthorHolliday, Nicholas D., AuthorHoriuchi, Mastgugu, AuthorHoyer, Daniel, AuthorHunyady, Laszlo, AuthorHusain, Ahsan, AuthorIJzerman, Adriaan P., AuthorInagami, Tadashi, AuthorJacobson, Kenneth A., AuthorJensen, Robert T., AuthorJockers, Ralf, AuthorJonnalagadda, Deepa, AuthorKarnik, Sadashiva, AuthorKaupmann, Klemens, AuthorKemp, Jacqueline, AuthorKennedy, Charles, AuthorKihara, Yasuyuki, AuthorKitazawa, Takio, AuthorKozielewicz, Pawel, AuthorKreienkamp, Hans-Juergen, AuthorKukkonen, Jyrki P., AuthorLangenhan, Tobias, AuthorLeach, Katie, AuthorLecca, Davide, AuthorLee, John D., AuthorLeeman, Susan E., AuthorLeprince, Jerome, AuthorLi, Xaria X., AuthorWilliams, Tom Lloyd, AuthorLolait, Stephen J., AuthorLupp, Amelie, AuthorMacrae, Robyn, AuthorMaguire, Janet, AuthorMazella, Jean, AuthorMcArdle, Craig A., AuthorMelmed, Shlomo, AuthorMichel, Martin C., AuthorMiller, Laurence J., AuthorMitolo, Vincenzo, AuthorMouillac, Bernard, AuthorMueller, Christa E., AuthorMurphy, Philip, AuthorNahon, Jean-Louis, AuthorNgo, Tony, AuthorNorel, Xavier, AuthorNyimanu, Duuamene, AuthorOcarroll, Anne-Marie, AuthorOffermanns, Stefan1, Author              Panaro, Maria Antonietta, AuthorParmentier, Marc, AuthorPertwee, Roger G., AuthorPin, Jean-Philippe, AuthorProssnitz, Eric R., AuthorQuinn, Mark, AuthorRamachandran, Rithwik, AuthorRay, Manisha, AuthorReinscheid, Rainer K., AuthorRondard, Philippe, AuthorRovati, G. Enrico, AuthorRuzza, Chiara, AuthorSanger, Gareth J., AuthorSchoeneberg, Torsten, AuthorSchulte, Gunnar, AuthorSchulz, Stefan, AuthorSegaloff, Deborah L., AuthorSerhan, Charles N., AuthorStoddart, Leigh A., AuthorSugimoto, Yukihiko, AuthorSummers, Roger, AuthorTan, Valerie P., AuthorThal, David, AuthorThomas, Walter (Wally), AuthorTimmermans, PieterB M. W. M., AuthorTirupula, Kalyan, AuthorTulipano, Giovanni, AuthorUnal, Hamiyet, AuthorUnger, Thomas, AuthorValant, Celine, AuthorVanderheyden, Patrick, AuthorVaudry, David, AuthorVaudry, Hubert, AuthorVilardaga, Jean-Pierre, AuthorWalker, Christopher S., AuthorWang, Ji Ming, AuthorWard, Donald T., AuthorWester, Hans-Juergen, AuthorWillars, Gary B., AuthorWoodruff, Trent M., AuthorYao, Chengcan, AuthorYe, Richard D., Author more..
1Pharmacology, Max Planck Institute for Heart and Lung Research, Max Planck Society, Ludwigstr. 43, D-61231 Bad Nauheim , DE, ou_2591696              


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 Abstract: The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at . G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.


 Dates: 2021-09-162021-10
 Publication Status: Published in print
 Pages: -
 Publishing info: -
 Table of Contents: -
 Rev. Type: -
 Identifiers: ISI: 000696321000003
DOI: 10.1111/bph.15538
PMID: 34529832
 Degree: -



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Source Genre: Journal
Publ. Info: -
Pages: - Volume / Issue: 178 (Supplement 1) Sequence Number: - Start / End Page: S27 - S156 Identifier: ISSN: 0007-1188