Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced 
Associate Domain Central Pocket

Karatas, Hacer; Akbarzadeh, Mohammad; Adihou, Hélène; Hahne, Gernot; Pobbati, Ajaybabu V.; Yihui Ng, Elizabeth; Guéret, Stéphanie M.; Sievers, Sonja; Pahl, Axel; Metz, Malte; Zinken, Sarah; Dötsch, Lara; Nowak, Christine; Thavam, Sasikala; Friese, Alexandra; Kang, CongBao; Hong, Wanjin; Waldmann, Herbert

doi:10.1021/acs.jmedchem.0c01275

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Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced Associate Domain Central Pocket

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/persons/resource/persons239234

Karatas, Hacer
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons243058

Akbarzadeh, Mohammad
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons202642

Adihou, Hélène
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons118867

Hahne, Gernot
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons202639

Guéret, Stéphanie M.
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons118736

Sievers, Sonja
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons198279

Pahl, Axel
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons202224

Metz, Malte
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons231959

Zinken, Sarah
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons226558

Dötsch, Lara
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons251191

Nowak, Christine
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons214421

Thavam, Sasikala
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons123083

Friese, Alexandra
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

/persons/resource/persons98735

Waldmann, Herbert
Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society;

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Citation

Karatas, H., Akbarzadeh, M., Adihou, H., Hahne, G., Pobbati, A. V., Yihui Ng, E., et al. (2020). Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced Associate Domain Central Pocket. Journal of Medicinal Chemistry, 63(20), 11972-11989. doi:10.1021/acs.jmedchem.0c01275.

Cite as: https://hdl.handle.net/21.11116/0000-0007-1D22-3

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